SCHEMBL21023784

SCHEMBL21023784

CC(C)c1cc(C(F)(F)F)nn1C1CCN(O)CC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.36
TGFBR1 P36897 4/20 0.33
TRPV1 Q8NER1 1/20 0.32
MAP3K12 Q12852 1/20 0.32
GAA P10253 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19105611 0.90 TGFBR1 (0.35) NR3C2TGFBR1TRPV1MAP3K12GAA
SCHEMBL19954525 0.89 SMN1; SMN2 (0.37) NR3C2TGFBR1MAP3K12GAAALDH1A1
SCHEMBL19954566 0.87 NR3C1 (0.36) NR3C2TGFBR1MAP3K12ALDH1A1
SCHEMBL19954663 0.87 NR3C2 (0.38) NR3C2TGFBR1TRPV1MAP3K12GAA
SCHEMBL19954553 0.87 NR3C2 (0.40) NR3C2TGFBR1TRPV1MAP3K12GAA
SCHEMBL19954523 0.86 TGFBR1 (0.35) NR3C2TGFBR1TRPV1MAP3K12
SCHEMBL21024127 0.85 NR3C2 (0.40) NR3C2TGFBR1TRPV1MAP3K12GAA
SCHEMBL19954664 0.84 MAPK1 (0.39) NR3C2TGFBR1TRPV1LMNAALDH1A1
SCHEMBL19954599 0.83 NR3C2 (0.39) NR3C2GAAALDH1A1MAPTTHRB
SCHEMBL19954637 0.83 ALDH1A1 (0.34) NR3C2MAP3K12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080087-B1 N-SUBSTITUTED PYRAZOLYL GUANIDINE F1F0-ATPASE INHIBITORS AND THERAPEUTIC USES THEREOF LYCERA CORP (US) 2019-05-22 EP disclosed