SCHEMBL21033908

SCHEMBL21033908

Fc1cc2nc(CC3CCCCC3)[nH]c2cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.53
IDO1 P14902 5/20 0.53
CACNA1H O95180 3/20 0.51
CACNA1G O43497 2/20 0.47
CACNA1C Q13936 1/20 0.47
OPRL1 P41146 1/20 0.44
F10 P00742 1/20 0.43
PDE10A Q9Y233 1/20 0.43
TXN P10599 1/20 0.42
GRIN1 Q05586 3/20 0.40
GRIN2B Q13224 3/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1255527 0.81 CACNA1H (0.43) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL21034171 0.81 MEN1 (0.57) AAK1IDO1CACNA1HCACNA1GCACNA1C
Hydrochloric Acid SCHEMBL1512918 0.80 CACNA1H (0.42) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL1257016 0.80 CACNA1H (0.44) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL21034664 0.78 AAK1 (0.50) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL21034692 0.76 IDO1 (0.54) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL8809271 0.76 AAK1 (0.51) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL21034524 0.76 AAK1 (0.51) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL17516021 0.76 AAK1 (0.51) AAK1IDO1CACNA1HCACNA1GCACNA1C
SCHEMBL21035092 0.76 IDO1 (0.57) AAK1IDO1CACNA1HCACNA1GCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019101188-A1 NOVEL BENZOIMIDAZOLES AS SELECTIVE INHIBITORS OF INDOLEAMINE 2, 3-DIOXYGENASES BEIGENE, LTD. (GB) 2019-05-31 WO disclosed