SCHEMBL21034664

SCHEMBL21034664

c1c2c(cc3[nH]c(CC4CCCCC4)nc13)OCO2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.50
PDE10A Q9Y233 1/20 0.48
CACNA1H O95180 3/20 0.45
CACNA1G O43497 2/20 0.43
CACNA1C Q13936 1/20 0.41
IDO1 P14902 4/20 0.39
BRS3 P32247 4/20 0.39
TPH1 P17752 2/20 0.39
TPH2 Q8IWU9 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PDE9A O76083 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CDC7 O00311 1/20 0.36
CCNE1 P24864 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21034171 0.78 MEN1 (0.57) AAK1PDE10ACACNA1HCACNA1GCACNA1C
SCHEMBL21033908 0.78 AAK1 (0.53) AAK1PDE10ACACNA1HCACNA1GCACNA1C
SCHEMBL12111153 0.77 GAA (0.56) PDE10ABRS3TPH1TPH2ALDH1A1
SCHEMBL6941291 0.74 PDE10A (0.50) PDE10ACACNA1GBRS3TPH1TPH2
Hydrochloric Acid SCHEMBL27136123 0.74 PDE10A (0.56) PDE10ACACNA1HIDO1BRS3TPH1
SCHEMBL21034524 0.72 AAK1 (0.51) AAK1CACNA1HCACNA1GCACNA1CIDO1
SCHEMBL8809271 0.72 AAK1 (0.51) AAK1CACNA1HCACNA1GCACNA1CIDO1
SCHEMBL17516021 0.72 AAK1 (0.51) AAK1CACNA1HCACNA1GCACNA1CIDO1
SCHEMBL21034692 0.72 IDO1 (0.54) AAK1CACNA1HCACNA1GCACNA1CIDO1
SCHEMBL21034172 0.71 IDO1 (0.57) AAK1CACNA1HCACNA1GCACNA1CIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019101188-A1 NOVEL BENZOIMIDAZOLES AS SELECTIVE INHIBITORS OF INDOLEAMINE 2, 3-DIOXYGENASES BEIGENE, LTD. (GB) 2019-05-31 WO disclosed