SCHEMBL21034976

SCHEMBL21034976

NC1CC2CCC(C1)C2C(=O)[C@@H]1C[C@H](Oc2ccc(Cl)c(-c3ccccc3)c2)CN1S(=O)(=O)c1ccc2cc(OC3CCCC3)ccc2c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.39
MMP9 P14780 4/20 0.38
CA12 O43570 2/20 0.35
CA2 P00918 2/20 0.35
MMP2 P08253 1/20 0.35
AKR1C3 P42330 6/20 0.34
AKR1C1 Q04828 2/20 0.34
HRH1 P35367 2/20 0.33
CCR3 P51677 2/20 0.33
KCNH2 Q12809 2/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
FFAR4 Q5NUL3 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21035658 1.00 GHSR (0.39) GHSRMMP9CA12CA2MMP2
SCHEMBL21035524 0.90 KAT6A (0.38) GHSRMMP9MMP2AKR1C3AKR1C1
SCHEMBL21034975 0.88 MMP9 (0.43) GHSRMMP9CA12CA2MMP2
SCHEMBL21035657 0.88 MMP9 (0.43) GHSRMMP9CA12CA2MMP2
SCHEMBL21035656 0.86 MCL1 (0.37) MMP9CA12CA2MMP2
Trifluoroacetic Acid SCHEMBL21002047 0.83 GHSR (0.40) GHSRMMP9CA12CA2MMP2
SCHEMBL21035353 0.78 GHSR (0.43) GHSRMMP9CA12CA2MMP2
SCHEMBL21034980 0.78 GHSR (0.43) GHSRMMP9CA12CA2MMP2
SCHEMBL21034984 0.77 CA12 (0.48) GHSRMMP9CA12CA2MMP2
SCHEMBL21035346 0.77 CA12 (0.48) GHSRMMP9CA12CA2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed