SCHEMBL21035486

SCHEMBL21035486

CC(C)(C)OC(=O)NC1CCN(C(=O)[C@@H]2CN(Cc3ccc(C4(C(F)(F)F)CC4)cc3)CCN2S(=O)(=O)c2ccc(OCC3CCCCC3)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 11/20 0.39
MMP1 P03956 11/20 0.39
MMP9 P14780 7/20 0.39
MMP3 P08254 3/20 0.39
MMP7 P09237 3/20 0.39
ADAM17 P78536 6/20 0.37
NAMPT P43490 1/20 0.37
ACACB O00763 1/20 0.37
CCR4 P51679 1/20 0.35
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21036241 1.00 MMP13 (0.39) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035620 0.97 MMP13 (0.38) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035357 0.91 MMP1 (0.38) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035570 0.91 MMP1 (0.40) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035604 0.89 SCN9A (0.39) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035503 0.89 EPHX2 (0.39) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21034944 0.89 PRKAA2 (0.40) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035340 0.88 MEN1 (0.41) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035442 0.88 MEN1 (0.41) MMP13MMP1MMP9MMP3MMP7
SCHEMBL21035600 0.88 MEN1 (0.41) MMP13MMP1MMP9MMP3MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed