SCHEMBL21035835

SCHEMBL21035835

CCC(=O)N[C@@H](CC(C)(C)C)C(=O)N1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.39
AURKA O14965 1/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39
PRKD3 O94806 1/20 0.39
PAK4 O96013 1/20 0.39
ABL1 P00519 1/20 0.39
NTRK1 P04629 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39
IGF1R P08069 1/20 0.39
MET P08581 1/20 0.39
PDGFRB P09619 1/20 0.39
PIM1 P11309 1/20 0.39
FGFR1 P11362 1/20 0.39
PDGFRA P16234 1/20 0.39
PRKACA P17612 1/20 0.39
LTK P29376 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21124133 0.85 CYP3A4 (0.41) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL21036085 0.85 SIGMAR1 (0.37) SIGMAR1CHRM5CHRM3ITGB3ITGA2B
SCHEMBL17011282 0.82 SIGMAR1 (0.37) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL16748082 0.82 SIGMAR1 (0.39) SIGMAR1CHRM5CHRM3ITGB3ITGA2B
SCHEMBL22303730 0.75 ITGB3 (0.45) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL14683864 0.73 HPGD (0.41) SIGMAR1CHRM5CHRM3HPGDCHRNB2
SCHEMBL16748054 0.73 HPGD (0.41) SIGMAR1CHRM5CHRM3HPGDCHRNB2
SCHEMBL16767821 0.72 DPP4 (0.48) SIGMAR1CHRM5CHRM3HPGDCHRNB2
SCHEMBL16745496 0.72 HPGD (0.40) SIGMAR1CHRM5CHRM3HPGDCHRNB2
SCHEMBL20994238 0.71 CYP3A4 (0.40) ITGB3ITGA2BUGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489231-B1 PIPERAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2021-06-09 EP disclosed
EP-3489231-A1 PIPERAZINE DERIVATIVE Astellas Pharma Inc. (JP) 2019-05-29 EP disclosed