SCHEMBL21044221

SCHEMBL21044221

COC(=O)c1cc(-c2cccc(Cl)c2)cc(C(=O)OC)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.52
SLC6A2 P23975 1/20 0.51
CNR2 P34972 3/20 0.48
TP53 P04637 2/20 0.45
MRGPRX4 Q96LA9 1/20 0.45
GRM5 P41594 1/20 0.45
CYP1A2 P05177 2/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
RECQL P46063 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PLA2G2A P14555 1/20 0.44
ABL1 P00519 1/20 0.44
VEGFA P15692 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1937391 0.86 CNR2 (0.59) SLC6A3SLC6A2CNR2TP53MRGPRX4
SCHEMBL21044529 0.83 SMN1; SMN2 (0.49) TP53CYP1A2MAPTNPC1SMN1; SMN2
SCHEMBL4592907 0.82 CNR2 (0.65) SLC6A3CNR2
SCHEMBL19915788 0.82 ALDH1A1 (0.55) CYP1A2MAPTSMN1; SMN2GAARECQL
SCHEMBL1938088 0.81 CNR2 (0.49) SLC6A3SLC6A2CNR2MRGPRX4PLA2G2A
SCHEMBL9034755 0.81 MAPK1 (0.48) TP53CYP1A2MAPTNPC1SMN1; SMN2
SCHEMBL3511154 0.81 SLC6A3 (0.55) SLC6A3SLC6A2MAPTNPC1SMN1; SMN2
SCHEMBL17595088 0.80 KMO (0.58) CNR2NPC1RAB9AL3MBTL1EGLN1
SCHEMBL7827008 0.79 PLAU (0.59) SLC6A3SLC6A2MAPTNPC1RAB9A
SCHEMBL24994712 0.79 CNR2 (0.52) SLC6A3SLC6A2CNR2MRGPRX4ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191451-B1 4-SUBSTITUTED PYRIDINE-2,6-DICARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING SAME OKINAWA INST SCIENCE & TECH SCHOOL CORP (JP) 2019-06-05 EP claimed