SCHEMBL21048952

SCHEMBL21048952

COc1ccc(CO[C@]2(c3ccc(Cl)cc3F)CC[C@]3(CC2)CO3)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.36
CTSD P07339 3/20 0.36
ALDH1A1 P00352 5/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
KCNA5 P22460 1/20 0.35
CNR1 P21554 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
XBP1 P17861 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17543027 1.00 BACE1 (0.36) BACE1CTSDALDH1A1HPGDKDM4E
SCHEMBL17543058 1.00 BACE1 (0.36) BACE1CTSDALDH1A1HPGDKDM4E
SCHEMBL17543986 0.88 ALDH1A1 (0.38) ALDH1A1HPGDKDM4ELMNAMAPT
SCHEMBL17543517 0.84 MEN1 (0.37) ALDH1A1MAPTKCNA5CNR1MAOA
SCHEMBL21048971 0.83 KCNA5 (0.37) ALDH1A1LMNAMAPTKCNA5CNR1
SCHEMBL17542690 0.83 KCNA5 (0.41) ALDH1A1MAPTKCNA5CNR1MAOA
SCHEMBL17542840 0.83 KCNA5 (0.37) ALDH1A1LMNAKCNA5CNR1MAOA
SCHEMBL17543118 0.80 BACE1 (0.36) BACE1CTSDALDH1A1SMN1; SMN2
SCHEMBL17543119 0.80 BACE1 (0.36) BACE1CTSDALDH1A1SMN1; SMN2
SCHEMBL17542733 0.75 KEAP1 (0.36) ALDH1A1LMNAHTTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3186240-B1 HETEROBICYCLIC COMPOUNDS AND THEIR USE FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2019-06-12 EP disclosed