Wiskostatin

Wiskostatin

SCHEMBL21067493

CN(C)C[C@H](O)Cn1c2ccc(Br)cc2c2cc(Br)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DNM1 Q05193 9/20 1.00
MAPT P10636 4/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
P2RX3 P56373 1/20 0.68
BAX Q07812 1/20 0.56
TP53 P04637 2/20 0.54
MAPK1 P28482 2/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX15 P16050 1/20 0.54
HTT P42858 3/20 0.54
NPSR1 Q6W5P4 3/20 0.54
LMNA P02545 2/20 0.54
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
RAD52 P43351 1/20 0.52
PER2 O15055 3/20 0.50
CRY1 Q16526 3/20 0.50
CRY2 Q49AN0 3/20 0.50
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Wiskostatin SCHEMBL5800361 1.00 DNM1 (1.00) DNM1MAPTSMN1; SMN2P2RX3BAX
Wiskostatin SCHEMBL29911343 1.00 DNM1 (1.00) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL410834 0.85 DNM1 (0.73) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL22830722 0.85 P2RX3 (0.76) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL21467809 0.83 DNM1 (0.71) DNM1MAPTSMN1; SMN2P2RX3PER2
SCHEMBL15592978 0.83 DNM1 (0.70) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL15880984 0.82 DNM1 (0.69) DNM1MAPTSMN1; SMN2HTTNPSR1
SCHEMBL25076450 0.81 P2RX3 (1.00) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL12013711 0.81 DNM1 (0.68) DNM1MAPTSMN1; SMN2P2RX3BAX
SCHEMBL30267744 0.81 DNM1 (0.68) DNM1MAPTSMN1; SMN2P2RX3BAX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11446398-B2 Regulated biocircuit systems OBSIDIAN THERAPEUTICS, INC. (US) 2022-09-20 US disclosed
US-20190192691-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. 2019-06-27 US disclosed