SCHEMBL210682

SCHEMBL210682

COC(=O)c1ccc(CNc2cc(Cl)nc(SC)n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
PTGES O14684 3/20 0.46
ALOX5 P09917 2/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TP53 P04637 1/20 0.44
DRD2 P14416 1/20 0.44
TBXA2R P21731 1/20 0.44
GAA P10253 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HDAC1 Q13547 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
PTGS2 P35354 2/20 0.42
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28202910 0.83 CLK4 (0.47) LMNAGAAMEN1KMT2ASMN1; SMN2
SCHEMBL16012065 0.80 VNN1 (0.44) ALDH1A1LMNANPSR1DRD2TBXA2R
SCHEMBL12321866 0.79 MEN1 (0.53) ALDH1A1PTGESALOX5LMNAGAA
SCHEMBL23291926 0.78 ALDH1A1 (0.52) ALDH1A1CA1CA2LMNADRD2
SCHEMBL3717932 0.77 ALDH1A1 (0.57) ALDH1A1CA1CA2PTGS2PIK3CA
SCHEMBL14801946 0.76 CA1 (0.47) ALDH1A1CA1CA2LMNATSHR
SCHEMBL14801417 0.76 MEN1 (0.50) LMNATSHRNPSR1TP53GAA
SCHEMBL209726 0.76 ALDH1A1 (0.53) ALDH1A1CA1CA2LMNADRD2
SCHEMBL3711270 0.76 PIK3CA (0.61) ALDH1A1CA1CA2LMNADRD2
SCHEMBL17581215 0.73 VNN1 (0.48) ALDH1A1GAAMEN1KMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-20070213330-A1 Anticancer agents; antiproliferative agents METHYLGENE INC. (CA) 2007-09-13 US disclosed
US-20070213330-A1 Anticancer agents; antiproliferative agents METHYLGENE INC. (CA) 2007-09-13 US disclosed
US-20070213330-A1 Anticancer agents; antiproliferative agents METHYLGENE INC. (CA) 2007-09-13 US disclosed
US-7253204-B2 Antiproliferative agents METHYLGENE INC. (CA) 2007-08-07 US disclosed
US-7253204-B2 Antiproliferative agents METHYLGENE INC. (CA) 2007-08-07 US disclosed
US-7253204-B2 Antiproliferative agents METHYLGENE INC. (CA) 2007-08-07 US disclosed
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP disclosed
US-20050245518-A1 Antiproliferative agents METHYLGENE, INC. 2005-11-03 US disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213330-A1 Anticancer agents; antiproliferative agents HDAC1, HDAC11, HDAC5 ALDH1A1 680/4885PTGES 4209/4885ALOX5 3601/4885
US-20050245518-A1 Antiproliferative agents HDAC1, HDAC11, HDAC5 ALDH1A1 758/4885PTGES 4133/4885ALOX5 3075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.