SCHEMBL3711270

SCHEMBL3711270

COC(=O)c1cc(Cl)nc(NCc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.61
PIK3CB P42338 1/20 0.61
ALDH1A1 P00352 2/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
PTGS2 P35354 1/20 0.52
F2 P00734 1/20 0.48
HIF1A Q16665 2/20 0.48
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
PAK4 O96013 1/20 0.47
ABL1 P00519 1/20 0.47
LCK P06239 1/20 0.47
FYN P06241 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
IGF1R P08069 1/20 0.47
PDGFRB P09619 1/20 0.47
FGFR1 P11362 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443320 0.87 HCAR2 (0.55) PIK3CAPIK3CBALDH1A1PTGS2AURKA
SCHEMBL3717932 0.87 ALDH1A1 (0.57) PIK3CAPIK3CBALDH1A1CA1CA2
SCHEMBL441290 0.84 PIK3CA (0.59) PIK3CAPIK3CBALDH1A1CA1CA2
SCHEMBL3716917 0.80 PIK3CA (0.52) PIK3CAPIK3CBALDH1A1CA1CA2
SCHEMBL3715503 0.79 PPARA (0.51) ALDH1A1HPGDKDM4E
SCHEMBL730969 0.77 LMNA (0.59) ALDH1A1HPGDKDM4ELMNA
SCHEMBL30931811 0.77 LMNA (0.59) ALDH1A1HPGDKDM4ELMNA
SCHEMBL29893730 0.77 CA1 (0.51) ALDH1A1CA1CA2F2KDM4E
SCHEMBL14842053 0.77 NOS2 (0.58) ALDH1A1PTGS2AURKADAPK3JAK2
SCHEMBL2135021 0.76 CA1 (0.47) ALDH1A1CA1CA2F2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed