SCHEMBL210703

SCHEMBL210703

Nc1ccccc1NC(=O)c1ccc2nc(-c3ccc(OC(F)(F)F)cc3)sc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.53
MAPT P10636 4/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TP53 P04637 2/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
KDM4E B2RXH2 2/20 0.47
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MITF O75030 1/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
RECQL P46063 1/20 0.47
GFER P55789 1/20 0.47
PAX8 Q06710 1/20 0.47
KLF5 Q13887 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211214 0.85 HDAC1 (0.74) HDAC1HDAC2HDAC3HDAC8CSNK2A2
SCHEMBL5583353 0.80 SMN1; SMN2 (0.65) HDAC1MAPTSMN1; SMN2TP53NPC1
SCHEMBL2091539 0.72 RORC (0.57) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL1988015 0.72 APP (0.69) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL22389485 0.72 RAB9A (0.66) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL15271195 0.72 SCD (0.74) HDAC1MAPTSMN1; SMN2TP53NPC1
SCHEMBL3947598 0.72 NPC1 (0.62) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL2192719 0.72 NPC1 (0.54) MAPTTP53NPC1RAB9AHDAC6
SCHEMBL2733518 0.71 HDAC1 (0.58) HDAC1CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL30795308 0.71 SCD (0.73) HDAC1MAPTSMN1; SMN2TP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed