SCHEMBL21075596

SCHEMBL21075596

CC(C)C1CCN(Cc2cc(Cl)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.42
CACNA1I Q9P0X4 1/20 0.42
CYP2D6 P10635 2/20 0.41
CYP3A4 P08684 1/20 0.41
USP2 O75604 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
FAAH O00519 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
UBE2M P61081 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
CXCR3 P49682 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
DDR1 Q08345 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21075227 0.86 L3MBTL1 (0.53) KCNH2CACNA1IL3MBTL1ACHEKDM4E
SCHEMBL19083894 0.85 ACHE (0.50) KCNH2CACNA1ICYP2D6CYP3A4USP2
SCHEMBL19075613 0.83 MGAT2 (0.45) KCNH2CACNA1ICYP2D6CYP3A4USP2
SCHEMBL19075615 0.78 CYP2D6 (0.49) KCNH2CYP2D6CYP3A4USP2CYP1A2
SCHEMBL19084132 0.77 CYP2D6 (0.51) KCNH2CYP2D6CYP3A4USP2CYP1A2
SCHEMBL19075643 0.77 RORC (0.42) KDM4EALDH1A1DCUN1D1TACR1
SCHEMBL19083685 0.76 CYP2D6 (0.52) KCNH2CYP2D6CYP3A4USP2CYP1A2
SCHEMBL19075619 0.75 SLC6A2 (0.47) KDM4EALDH1A1DCUN1D1
SCHEMBL23118445 0.74 CYP2D6 (0.50) KCNH2CYP2D6CYP3A4USP2CYP1A2
SCHEMBL20697685 0.74 ALOX5AP (0.44) UBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166939-B1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH INC (US) 2019-06-05 EP disclosed