SCHEMBL21075678

SCHEMBL21075678

NC1CCN(Cc2cc(C(F)(F)F)cc(C3CC3)n2)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.43
SLC6A4 P31645 7/20 0.43
KCNH2 Q12809 7/20 0.43
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
GRM2 Q14416 3/20 0.36
DRD4 P21917 3/20 0.36
DRD2 P14416 2/20 0.36
ADORA1 P30542 2/20 0.36
IDH2 P48735 1/20 0.36
HTT P42858 1/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19083939 0.87 TACR1 (0.45) TACR1SLC6A4KCNH2GRM2DRD4
SCHEMBL21075333 0.86 KCNH2 (0.44) TACR1SLC6A4KCNH2SIGMAR1
SCHEMBL19075523 0.85 KCNH2 (0.44) TACR1SLC6A4KCNH2GRM2DRD4
SCHEMBL21075802 0.84 TACR1 (0.49) TACR1SLC6A4KCNH2
SCHEMBL6945302 0.74 CYP2D6 (0.52) SIGMAR1
SCHEMBL17061916 0.74 TACR1 (0.46) TACR1SLC6A4KCNH2
SCHEMBL16770692 0.74 TACR1 (0.46) TACR1SLC6A4KCNH2
SCHEMBL4023227 0.73 KCNH2 (0.45) TACR1SLC6A4KCNH2
SCHEMBL4021955 0.73 TACR1 (0.45) TACR1SLC6A4KCNH2GRM2
SCHEMBL17069228 0.71 TACR1 (0.44) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166939-B1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH INC (US) 2019-06-05 EP disclosed