SCHEMBL21077808

SCHEMBL21077808

OC1(c2ccccc2Cl)CCN(I)CC1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.49
DRD4 P21917 2/20 0.49
DRD3 P35462 2/20 0.49
OPRL1 P41146 13/20 0.45
OPRM1 P35372 12/20 0.45
OPRD1 P41143 12/20 0.45
OPRK1 P41145 12/20 0.45
PKLR P30613 2/20 0.40
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16565590 0.82 OPRL1 (0.51) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL27035066 0.79 HDAC4 (0.49) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL17886563 0.78 OPRM1 (0.47) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL8986019 0.77 HDAC4 (0.51) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL30089861 0.77 HDAC4 (0.51) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL23210134 0.74 OPRM1 (0.44) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL29691231 0.74 OPRM1 (0.44) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL652087 0.74 SIGMAR1 (0.57) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL7109502 0.73 DRD2 (0.54) DRD2DRD4DRD3OPRL1OPRM1
SCHEMBL7237487 0.73 DRD2 (0.60) DRD2DRD4DRD3OPRL1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed