SCHEMBL21077975

SCHEMBL21077975

CCc1ccc(C(=O)NCc2cncc(C)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.53
HDAC1 Q13547 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.51
LMNA P02545 2/20 0.51
POLB P06746 2/20 0.51
HPGD P15428 2/20 0.51
GLA P06280 1/20 0.51
MAPK1 P28482 1/20 0.50
NLRP1 Q9C000 1/20 0.50
KDM1A O60341 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MMP13 P45452 1/20 0.49
TRPV1 Q8NER1 1/20 0.49
NAMPT P43490 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17888293 0.90 HDAC1 (0.60) PIK3CAHDAC1SMN1; SMN2LMNAPOLB
SCHEMBL19226518 0.85 LMNA (0.66) LMNAMEN1KMT2ANAMPTCYP1A2
SCHEMBL19226517 0.84 SMN1; SMN2 (0.59) PIK3CAHDAC1SMN1; SMN2LMNAPOLB
SCHEMBL18617541 0.82 TRPV1 (0.53) PIK3CAHDAC1SMN1; SMN2LMNAPOLB
SCHEMBL27220658 0.82 EPHX2 (0.61) SMN1; SMN2LMNAHPGDMAPK1MMP13
SCHEMBL21214344 0.82 PIK3CA (0.48) PIK3CAHDAC1SMN1; SMN2LMNAPOLB
SCHEMBL10076246 0.79 TRPV1 (0.74) SMN1; SMN2LMNAPOLBHPGDGLA
SCHEMBL12058757 0.78 LMNA (0.69) SMN1; SMN2LMNAPOLBHPGDMAPK1
SCHEMBL19322933 0.76 CYP2C9 (0.48) PIK3CANAMPTCYP2C9GAAMAPT
SCHEMBL8374098 0.76 L3MBTL1 (0.71) SMN1; SMN2LMNAPOLBHPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed