SCHEMBL21078014

SCHEMBL21078014

CC(=O)NCC1(c2ccc(Cl)cc2)CCN(I)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.56
DRD2 P14416 1/20 0.56
DRD4 P21917 1/20 0.56
P2RX7 Q99572 10/20 0.53
MCHR1 Q99705 3/20 0.47
CNR1 P21554 1/20 0.47
TSHR P16473 1/20 0.45
CASP1 P29466 1/20 0.45
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16565532 0.88 P2RX7 (0.67) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL21214320 0.84 DRD3 (0.54) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL20004196 0.84 DRD2 (0.54) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL16553711 0.81 DRD2 (0.53) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL16554105 0.79 DRD2 (0.50) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL28077553 0.79 DRD2 (0.50) DRD3DRD2DRD4P2RX7MCHR1
SCHEMBL21078155 0.77 EPHX2 (0.43) DRD3DRD2DRD4P2RX7SLC6A2
SCHEMBL21078008 0.76 DRD2 (0.49) DRD3DRD2DRD4P2RX7SLC6A2
SCHEMBL21078137 0.76 SLC6A4 (0.41) DRD2P2RX7SLC6A4SLC6A3
SCHEMBL11602483 0.75 DRD4 (0.55) DRD3DRD2DRD4P2RX7CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed