SCHEMBL28077553

SCHEMBL28077553

CC(=O)NCC1(c2ccc(Cl)cc2)CCN(OC(=O)C(C)(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.50
DRD3 P35462 2/20 0.50
DRD4 P21917 1/20 0.50
P2RX7 Q99572 7/20 0.47
TSHR P16473 1/20 0.42
CASP1 P29466 1/20 0.42
MCHR1 Q99705 2/20 0.42
CNR1 P21554 1/20 0.41
KCNH2 Q12809 1/20 0.39
CACNA1I Q9P0X4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20004196 0.84 DRD2 (0.54) DRD2DRD3DRD4P2RX7TSHR
SCHEMBL28831246 0.83 SLC6A4 (0.48) DRD2P2RX7
SCHEMBL16554105 0.82 DRD2 (0.50) DRD2DRD3DRD4P2RX7TSHR
SCHEMBL28077739 0.81 DRD2 (0.39) DRD2P2RX7CNR1
SCHEMBL28077613 0.81 DRD2 (0.39) DRD2P2RX7CNR1
SCHEMBL28077873 0.81 DRD2 (0.39) DRD2P2RX7CNR1
SCHEMBL16565532 0.80 P2RX7 (0.67) DRD2DRD3DRD4P2RX7MCHR1
SCHEMBL21078014 0.79 DRD3 (0.56) DRD2DRD3DRD4P2RX7TSHR
SCHEMBL28077607 0.79 EPHX2 (0.45) DRD2P2RX7CNR1
SCHEMBL373464 0.78 DRD3 (0.48) DRD2DRD3DRD4P2RX7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745209-A Triazolopyridine compounds, compositions, and methods of use thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed