SCHEMBL21078095

SCHEMBL21078095

O=C1N(I)C(c2ccccc2)C12CCNCC2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.37
SIGMAR1 Q99720 3/20 0.37
OPRM1 P35372 1/20 0.37
SLC18A3 Q16572 1/20 0.37
TSHR P16473 1/20 0.36
USP2 O75604 2/20 0.35
CYP2D6 P10635 2/20 0.35
KDM1A O60341 3/20 0.35
MAOB P27338 2/20 0.35
OPRD1 P41143 1/20 0.35
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
DRD2 P14416 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TRPV1 Q8NER1 2/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17888239 0.81 OPRK1 (0.38) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL8202443 0.80 TRPV1 (0.49) HSD17B10TSHRUSP2CYP2D6CYP3A4
SCHEMBL17886562 0.79 TRPV1 (0.36) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL21788683 0.78 TRPV1 (0.37) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL8212506 0.72 ALDH1A1 (0.43) HSD17B10TRPV1
SCHEMBL26669761 0.71 SLC18A3 (0.41) SIGMAR1SLC18A3KDM1AMAOBCYP3A4
SCHEMBL24621328 0.70 TSHR (0.40) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL18746129 0.69 MAPT (0.42) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL8202509 0.68 TSHR (0.41) HSD17B10SIGMAR1OPRM1SLC18A3TSHR
SCHEMBL1138335 0.67 SLC6A9 (0.56) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed