SCHEMBL21079055

SCHEMBL21079055

CC(C)C(=O)Nc1cc([C@H](C)N)ccn1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.50
RIOK2 Q9BVS4 4/20 0.44
MAPT P10636 6/20 0.44
GSK3B P49841 5/20 0.44
ACVRL1 P37023 1/20 0.44
POLB P06746 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAP4K1 Q92918 1/20 0.43
NR3C2 P08235 2/20 0.42
GSK3A P49840 2/20 0.41
MAPK10 P53779 2/20 0.41
BRAF P15056 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15358570 1.00 TYK2 (0.50) TYK2RIOK2MAPTGSK3BACVRL1
Hydrochloric Acid SCHEMBL15350070 0.98 TYK2 (0.49) TYK2RIOK2MAPTGSK3BACVRL1
SCHEMBL15627415 0.87 TYK2 (0.52) TYK2RIOK2MAPTGSK3BACVRL1
SCHEMBL27342084 0.86 TYK2 (0.51) TYK2RIOK2MAPTGSK3BACVRL1
SCHEMBL22809608 0.86 TYK2 (0.51) TYK2RIOK2MAPTGSK3BACVRL1
SCHEMBL15358566 0.86 AAK1 (0.49) TYK2
SCHEMBL21078952 0.86 AAK1 (0.49) TYK2
Hydrochloric Acid SCHEMBL15350524 0.84 AAK1 (0.48) TYK2
SCHEMBL25997633 0.82 TYK2 (0.48) TYK2RIOK2MAPTGSK3BACVRL1
SCHEMBL15358582 0.82 LMNA (0.45) MAPTGSK3BPOLBNR3C2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2841421-B1 AMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2019-06-05 EP disclosed