Mindodilol

Mindodilol

SCHEMBL2107921

OC(COc1cccc2[nH]ccc12)CN1CCC(COc2ccccc2)CC1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.63
ADRB1 P08588 1/20 0.63
ADRB3 P13945 1/20 0.63
HTR1A P08908 18/20 0.62
SLC6A4 P31645 4/20 0.62
DRD2 P14416 1/20 0.57
DRD4 P21917 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mindodilol SCHEMBL11540170 1.00 ADRB2 (0.63) ADRB2ADRB1ADRB3HTR1ASLC6A4
Mindodilol SCHEMBL6295415 0.95 ADRB2 (0.61) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL11541170 0.89 HTR1A (0.64) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL11541941 0.89 ADRB2 (0.59) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL11539522 0.89 HTR1A (0.66) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL7876327 0.88 DRD2 (0.74) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL11540486 0.88 ADRB2 (0.61) ADRB2ADRB1ADRB3HTR1ASLC6A4
Benzoic Acid SCHEMBL11544384 0.88 HTR1A (0.57) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL7885674 0.87 DRD4 (0.73) ADRB2ADRB1ADRB3HTR1ASLC6A4
SCHEMBL11537570 0.86 DRD4 (0.52) ADRB2ADRB1ADRB3HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 121 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-6852337-B2 Carvedilol-galenics ROCHE DIAGNOSTICS GMBH (DE) 2005-02-08 US claimed
EP-1069896-B1 CARVEDILOL-GALENICS ROCHE DIAGNOSTICS GMBH (DE) 2003-08-06 EP claimed
US-20030118643-A1 Carvedilol-galenics GABEL ROLF-DIETER (DE) 2003-06-26 US claimed
EP-1069896-A1 CARVEDILOL-GALENICS Roche Diagnostics GmbH (DE) 2001-01-24 EP claimed
US-4782043-A HYPOTENSIVES MERCK & CO., INC. (US) 1988-11-01 US claimed
EP-0278158-A2 Renin inhibitors containing phenylalanyl-histidine replacements MERCK & CO. INC. (US) 1988-08-17 EP claimed
EP-0273696-A2 Renin inhibitors containing histidine replacements MERCK & CO. INC. (US) 1988-07-06 EP claimed
EP-0209897-A2 Peptide enzyme inhibitors MERCK & CO. INC. (US) 1987-01-28 EP claimed
EP-0163237-A2 Di- and tri-peptidal renin inhibitors MERCK & CO. INC. (US) 1985-12-04 EP claimed
EP-0157409-A2 Renin inhibitors containing 2-substituted statine MERCK & CO. INC. (US) 1985-10-09 EP claimed
EP-0156318-A2 C-terminal amide cyclic renin inhibitors containing peptide isosteres MERCK & CO. INC. (US) 1985-10-02 EP claimed
EP-0156322-A2 Renin inhibitors containing peptide isosteres MERCK & CO. INC. (US) 1985-10-02 EP claimed
EP-0129189-A2 Renin inhibitors containing a C-terminal amide cycle and compositions and combinations containing the same MERCK & CO. INC. (US) 1984-12-27 EP claimed
US-4146630-A HYPOTENSIVE AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1979-03-27 US claimed