SCHEMBL21088010

SCHEMBL21088010

Nc1ccc(F)cc1-c1cc(F)cc(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
KEAP1 Q14145 1/20 0.41
CCNE2 O96020 2/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
BACE1 P56817 1/20 0.36
NPC1 O15118 1/20 0.36
CYP1A1 P04798 2/20 0.35
NOS3 P29474 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
MAP4K4 O95819 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ABL1 P00519 1/20 0.33
BRD4 O60885 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557724 0.84 ALDH1A1 (0.52) ALDH1A1KEAP1CCNE2CCNE1CDK2
SCHEMBL29901139 0.83 ALDH1A1 (0.62) ALDH1A1KEAP1CCNE2CCNE1CDK2
SCHEMBL21088009 0.83 ALDH1A1 (0.52) ALDH1A1KEAP1CCNE2CCNE1CDK2
SCHEMBL28228449 0.82 ALDH1A1 (0.44) ALDH1A1KEAP1TAAR1BACE1CYP1A1
Hydrochloric Acid SCHEMBL29901111 0.80 ALDH1A1 (0.59) ALDH1A1KEAP1CCNE2CCNE1CDK2
SCHEMBL3789841 0.80 TAAR1 (0.50) ALDH1A1KEAP1CCNE2CCNE1CDK2
SCHEMBL3793169 0.80 ALDH1A1 (0.54) ALDH1A1KEAP1TAAR1BACE1CYP1A2
SCHEMBL29492484 0.80 ALDH1A1 (0.54) ALDH1A1KEAP1TAAR1BACE1CYP1A2
Hydrochloric Acid SCHEMBL9311952 0.78 ALDH1A1 (0.52) ALDH1A1KEAP1TAAR1BACE1CYP1A2
Ammonia Solution, Strong SCHEMBL11901716 0.78 ALDH1A1 (0.52) ALDH1A1KEAP1TAAR1BACE1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019110521-A1 FLUOROPHENYL SUBSTITUTED MUSCARINIC RECEPTOR LIGANDS WITH SELECTIVITY FOR M3 OVER M2 Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2019-06-13 WO disclosed