SCHEMBL21088669

SCHEMBL21088669

NC(=O)C1CC1/C=C\c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.58
CTSK P43235 1/20 0.43
CYP1A2 P05177 2/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
PLIN1 O60240 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
RECQL P46063 2/20 0.41
PLIN5 Q00G26 2/20 0.41
ABHD5 Q8WTS1 2/20 0.41
TNKS O95271 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21088859 1.00 KDM1A (0.58) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL18172735 0.86 KDM1A (0.56) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL18173266 0.86 KDM1A (0.56) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL18172738 0.86 KDM1A (0.56) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL27799460 0.82 CTSK (0.59) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL21088922 0.80 KDM1A (0.50) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL18182909 0.80 KDM1A (0.50) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL21088849 0.79 KDM1A (0.49) KDM1ACTSKCYP1A2HDAC3HDAC4
SCHEMBL18172939 0.79 KDM1A (0.49) KDM1ACTSKCYP1A2LMNAMAPT
SCHEMBL18172936 0.79 KDM1A (0.49) KDM1ACTSKCYP1A2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed