SCHEMBL21089369

SCHEMBL21089369

CCCCc1ncc(C2CC2)cc1S(C)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
APLNR P35414 3/20 0.34
PTAFR P25105 1/20 0.34
NAAA Q02083 1/20 0.33
DRD2 P14416 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
TYK2 P29597 3/20 0.31
SPHK1 Q9NYA1 2/20 0.31
HDAC6 Q9UBN7 1/20 0.31
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196388 0.85 PTAFR (0.34) PTAFRDRD2SIGMAR1TYK2NR1H2
SCHEMBL17177879 0.74 TYK2 (0.42) TYK2NR1H2NR1H3
SCHEMBL18811516 0.74 PTAFR (0.33) PTAFRDRD2SIGMAR1TYK2
SCHEMBL21354998 0.73 MAP3K12 (0.43) TYK2NR1H2NR1H3
SCHEMBL17173652 0.72 TYK2 (0.34) TYK2NR1H2NR1H3
SCHEMBL24587299 0.71 LRRK2 (0.37) TYK2NR1H2NR1H3
SCHEMBL21089373 0.70 THRA (0.34) HDAC6NR1H2NR1H3
SCHEMBL23564201 0.70 SPHK1 (0.40) APLNRSPHK1
SCHEMBL20885627 0.69 TYK2 (0.34) TYK2
SCHEMBL17504812 0.69 KDM4E (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3495360-A1 HETEROARYL SUBSTITUTED HETEROCYCLYL SULFONES Grünenthal GmbH (DE) 2019-06-12 EP disclosed