SCHEMBL21091971

SCHEMBL21091971

CCNC(C)c1ccc(F)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.37
SLC6A4 P31645 5/20 0.35
SLC6A3 Q01959 4/20 0.35
CASR P41180 4/20 0.35
HTR2B P41595 2/20 0.33
GPR65 Q8IYL9 2/20 0.33
ADRA2C P18825 2/20 0.33
SLC6A2 P23975 2/20 0.33
HTR2C P28335 2/20 0.33
OPRM1 P35372 2/20 0.33
DRD3 P35462 2/20 0.33
HTR1B P28222 1/20 0.33
MLNR O43193 1/20 0.33
ABCB11 O95342 1/20 0.33
ADRB1 P08588 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2D6 P10635 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD2 P14416 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16849226 0.84 SIGMAR1 (0.40) SIGMAR1SLC6A4SLC6A3CASRHTR2B
SCHEMBL29198591 0.82 POLB (0.54) SIGMAR1CASRPOLB
SCHEMBL178501 0.80 SLC6A4 (0.39) SIGMAR1SLC6A4SLC6A3HTR2BGPR65
SCHEMBL12463310 0.75 HTR2B (0.42) SIGMAR1SLC6A4SLC6A3HTR2BGPR65
SCHEMBL28339998 0.75 CASR (0.56) SIGMAR1SLC6A4SLC6A3CASRHTR2B
SCHEMBL21091967 0.75 CASR (0.56) SIGMAR1SLC6A4SLC6A3CASRHTR2B
SCHEMBL13077642 0.75 CASR (0.56) SIGMAR1SLC6A4SLC6A3CASRHTR2B
SCHEMBL30488987 0.75 CASR (0.56) SIGMAR1SLC6A4SLC6A3CASRHTR2B
SCHEMBL10039768 0.72 CASR (0.73) CASR
SCHEMBL24017669 0.72 SIGMAR1 (0.37) SIGMAR1SLC6A4SLC6A3HTR2BGPR65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817299-B1 SUBSTITUTED CHROMAN COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS LUPIN LTD (IN) 2019-06-12 EP disclosed