Tazeprofen

Tazeprofen

SCHEMBL2109458

CC(C(=O)O)c1ccc2nc(-c3ccccc3)sc2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.62
KDM4E B2RXH2 6/20 0.62
NFKB1 P19838 5/20 0.62
NFKB2 Q00653 5/20 0.62
RELA Q04206 5/20 0.62
LMNA P02545 2/20 0.62
MAPT P10636 5/20 0.54
HPGD P15428 5/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
PKM P14618 4/20 0.54
ALDH1A1 P00352 3/20 0.54
GAA P10253 3/20 0.54
GLA P06280 1/20 0.54
RAB9A P51151 7/20 0.52
PAX8 Q06710 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
NOD2 Q9HC29 1/20 0.52
PTGS2 P35354 3/20 0.50
NPC1 O15118 6/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10939891 0.89 KDM4E (0.58) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL28868336 0.84 MAPT (0.68) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL13799598 0.80 LDHA (0.51) SMN1; SMN2MAPTHPGDMEN1KMT2A
SCHEMBL74053 0.79 RAB9A (0.68) SMN1; SMN2KDM4ELMNAMAPTHPGD
Cicloprofen SCHEMBL11060470 0.78 PTGS2 (0.46) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL121572 0.77 KDM4E (1.00) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL27682548 0.76 KDM4E (0.43) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL121577 0.76 KDM4E (0.81) SMN1; SMN2KDM4ENFKB1NFKB2RELA
SCHEMBL12565259 0.75 RAB9A (0.71) SMN1; SMN2KDM4EMAPTGAAGLA
SCHEMBL4132162 0.75 DYRK1A (0.63) SMN1; SMN2MEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-0017543-B1 BENZOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR THERAPEUTICAL USES Albert ROLLAND S.A. Société dite (FR) 1983-09-28 EP claimed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 US disclosed
US-10463611-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2019-11-05 US disclosed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US disclosed
US-20140154313-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2014-06-05 US disclosed
EP-2717860-A1 CONTROLLED ABSORPTION WATER-SOLUBLE PHARMACEUTICALLY ACTIVE ORGANIC COMPOUND FORMULATION FOR ONCE-DAILY ADMINISTRATION STI Pharma, LLC (US) 2014-04-16 EP disclosed
WO-1996039377-A1 FACE-TO-FACE/FACE-TO-EDGE INTERACTIVE CHIRAL SELECTORS AND RELATED APPARATUSES RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1996-12-12 WO disclosed
US-5484530-A CARBOXYLIC ACIDS AND ENANTIOMORPHS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1996-01-16 US disclosed
US-5387338-A An optical isomer separators RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1995-02-07 US disclosed
US-5256293-A Immobilizing enantiomer on support effective for use in chromatographic separation RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-10-26 US disclosed
WO-1993006080-A1 SEPARATION OF ENANTIOMERS OF NON-STEROIDAL ANTI-INFLAMMATORY DRUGS AND CHIRAL SELECTOR THEREFOR RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-04-01 WO disclosed
US-5028603-A Platelet-Activating Factor Antagonist; Useful In Treatment Of Inflammatory Diseases, Allergic Diseases, Asthma, Respiratory System Disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-07-02 US disclosed
EP-0316456-A1 ESTER-SUBSTITUTED THIENOTRIAZOLODIAZEPINE COMPOUNDS AND THEIR MEDICINAL USE Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-05-24 EP disclosed