SCHEMBL21096166

SCHEMBL21096166

O=C(Nc1ccc(F)cc1)c1ccc(OC(F)F)cn1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.56
LMNA P02545 1/20 0.56
RAB9A P51151 2/20 0.55
NPC1 O15118 1/20 0.55
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
P4HTM Q9NXG6 2/20 0.53
GRM4 Q14833 2/20 0.52
BACE1 P56817 9/20 0.51
MEN1 O00255 2/20 0.50
AGTR1 P30556 1/20 0.50
TLR9 Q9NR96 1/20 0.50
GSK3A P49840 1/20 0.49
GSK3B P49841 1/20 0.49
BACE2 Q9Y5Z0 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934432 0.83 SMN1; SMN2 (0.61) KMT2ALMNARAB9ANPC1ALDH1A1
SCHEMBL15886256 0.82 BACE1 (0.60) KMT2ARAB9ANPC1SMN1; SMN2GRM4
SCHEMBL6934524 0.82 NPC1 (0.56) KMT2ARAB9ANPC1ALDH1A1GAA
SCHEMBL6874915 0.80 NPC1 (0.69) KMT2ARAB9ANPC1ALDH1A1GAA
SCHEMBL21595576 0.78 SMN1; SMN2 (0.56) KMT2ARAB9ANPC1ALDH1A1GAA
SCHEMBL30763098 0.78 SMN1; SMN2 (0.56) KMT2ARAB9ANPC1ALDH1A1GAA
SCHEMBL4115554 0.77 MEN1 (0.59) KMT2ALMNARAB9ANPC1ALDH1A1
SCHEMBL17668487 0.77 LMNA (0.42) KMT2ALMNAP4HTMGRM4BACE1
SCHEMBL31277715 0.76 NPC1 (0.63) KMT2ARAB9ANPC1ALDH1A1GAA
SCHEMBL16006837 0.76 RAB9A (0.66) KMT2ALMNARAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855469-B1 5-AMINO[1,4]THIAZINES AS BACE 1 INHIBITORS HOFFMANN LA ROCHE (CH) 2019-06-19 EP disclosed