SCHEMBL211135

SCHEMBL211135

COC(=O)[C@@H](COC(=O)Nc1cc2ccccc2cn1)N(NCc1ccccc1Cl)C(C)=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
NOTUM Q6P988 1/20 0.37
CTSK P43235 1/20 0.36
HTT P42858 2/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
CSNK1D P48730 2/20 0.35
MAPK1 P28482 1/20 0.35
ABL1 P00519 5/20 0.35
WNT3A P56704 1/20 0.35
LMNA P02545 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL212597 0.93 NOTUM (0.37) ALDH1A1NOTUMCTSKNPC1SMN1; SMN2
SCHEMBL210077 0.87 NOTUM (0.36) ALDH1A1NOTUMCTSKHTTNPC1
SCHEMBL210644 0.86 NOTUM (0.36) ALDH1A1NOTUMCTSKNPC1CSNK1D
SCHEMBL212116 0.86 CTSK (0.36) ALDH1A1NOTUMCTSKHTTSMN1; SMN2
SCHEMBL212590 0.85 CTSK (0.36) ALDH1A1NOTUMCTSKCSNK1DABL1
SCHEMBL210694 0.84 NOTUM (0.34) ALDH1A1NOTUMCTSKHTTSMN1; SMN2
SCHEMBL211462 0.84 CTSK (0.36) ALDH1A1NOTUMCTSKHTTSMN1; SMN2
SCHEMBL2722110 0.84 ALDH1A1 (0.42) ALDH1A1NOTUMCTSKHTTNPC1
SCHEMBL4353508 0.84 CTSK (0.37) ALDH1A1NOTUMCTSKNPC1CSNK1D
SCHEMBL212341 0.83 CTSK (0.37) ALDH1A1NOTUMCTSKHTTCSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US claimed
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed