SCHEMBL21130686

SCHEMBL21130686

CN(CCc1ccccc1)C1(C)CCN(CCc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.53
SIGMAR1 Q99720 8/20 0.52
SLC6A3 Q01959 1/20 0.51
OPRM1 P35372 2/20 0.48
HTR1A P08908 1/20 0.46
DRD2 P14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970787 0.74 SLC6A3 (0.56) ACHESIGMAR1SLC6A3OPRM1HTR1A
SCHEMBL8970769 0.74 SLC6A3 (0.56) ACHESIGMAR1SLC6A3OPRM1HTR1A
SCHEMBL21726765 0.73 SLC6A3 (0.59) ACHESIGMAR1SLC6A3HTR1ADRD2
SCHEMBL6056974 0.73 SLC6A3 (0.83) ACHESIGMAR1SLC6A3HTR1ADRD2
SCHEMBL7264546 0.73 SLC6A3 (0.83) ACHESIGMAR1SLC6A3HTR1ADRD2
SCHEMBL14407778 0.73 SLC6A3 (0.83) ACHESIGMAR1SLC6A3HTR1ADRD2
SCHEMBL13150782 0.73 SLC6A3 (0.83) ACHESIGMAR1SLC6A3HTR1ADRD2
SCHEMBL3566447 0.73 SLC6A3 (0.54) ACHESIGMAR1SLC6A3OPRM1
SCHEMBL8970828 0.73 SIGMAR1 (0.56) ACHESIGMAR1SLC6A3OPRM1
SCHEMBL27638865 0.73 SLC6A3 (0.63) ACHESIGMAR1SLC6A3HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3221314-B1 SPIRO-ISOQUINOLINE-1,4'-PIPERIDINE COMPOUNDS HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS SA (ES) 2019-07-03 EP disclosed