SCHEMBL21135207

SCHEMBL21135207

C/C=N/Nc1cc2nc(C(=O)NC)cn2c(N2CCOCC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.41
PIK3CB P42338 1/20 0.40
NAPEPLD Q6IQ20 1/20 0.37
ALDH1A1 P00352 3/20 0.36
MAPT P10636 10/20 0.35
KDM4E B2RXH2 9/20 0.35
ATM Q13315 1/20 0.35
LMNA P02545 5/20 0.35
GAA P10253 4/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
TAAR1 Q96RJ0 2/20 0.35
APAF1 O14727 2/20 0.35
HTT P42858 1/20 0.35
MAPK10 P53779 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 4/20 0.35
NSD2 O96028 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21135206 0.89 ATR (0.38) ATRPIK3CBALDH1A1MAPTKDM4E
SCHEMBL21135204 0.87 PIK3CB (0.39) ATRPIK3CBALDH1A1MAPTKDM4E
SCHEMBL23272155 0.85 KDM4E (0.55) ATRALDH1A1MAPTKDM4EATM
SCHEMBL30312323 0.85 KDM4E (0.55) ATRALDH1A1MAPTKDM4EATM
SCHEMBL21135208 0.84 ATR (0.37) ATRPIK3CBALDH1A1MAPTKDM4E
SCHEMBL30312419 0.77 MAPT (0.57) ALDH1A1MAPTKDM4EATMLMNA
SCHEMBL21054975 0.77 MAPT (0.57) ALDH1A1MAPTKDM4EATMLMNA
SCHEMBL21135848 0.76 PIK3CA (0.51) PIK3CBALDH1A1MAPTKDM4ENPC1
SCHEMBL21135205 0.75 ATR (0.53) ATRNAPEPLDALDH1A1MAPTKDM4E
SCHEMBL23272117 0.75 KDM4E (0.57) ALDH1A1MAPTKDM4EATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019113523-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF BAJJI ASHOK (US) 2019-06-13 WO disclosed