SCHEMBL21152449

SCHEMBL21152449

C=N/N=C(/NN)c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
HPGD P15428 2/20 0.36
ERCC5 P28715 1/20 0.35
FEN1 P39748 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP2C9 P11712 1/20 0.33
POLB P06746 2/20 0.33
FFAR1 O14842 1/20 0.33
TYK2 P29597 1/20 0.33
MYC P01106 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13208833 0.79 MAOA (0.44) MAOAMAOBHPGDERCC5FEN1
SCHEMBL533919 0.72 SIGMAR1 (0.43) MAOAMAOBHPGDERCC5FEN1
SCHEMBL23416547 0.72 MAOA (0.37) MAOAMAOBHPGDERCC5FEN1
SCHEMBL17319502 0.70 ALDH1A1 (0.36) HPGDNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL20025577 0.69 MAOA (0.44) MAOAMAOBHPGDERCC5FEN1
SCHEMBL2992101 0.68 MAOA (0.41) MAOAMAOBHPGDERCC5FEN1
SCHEMBL2992104 0.68 MAOA (0.41) MAOAMAOBHPGDERCC5FEN1
SCHEMBL1128274 0.67 HPGD (0.60) MAOAMAOBHPGDERCC5FEN1
SCHEMBL3957272 0.67 MAOA (0.47) MAOAMAOBHPGDERCC5FEN1
SCHEMBL4749109 0.67 MAOA (0.47) MAOAMAOBHPGDERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2696878-B1 DOSAGE REGIMEN FOR SAPACITABINE AND DECITABINE IN COMBINATION FOR TREATING ACUTE MYELOID LEUKEMIA CYCLACEL LTD (GB) 2019-07-10 EP disclosed