SCHEMBL21152576

SCHEMBL21152576

C1=C(P(c2ccccc2)c2ccccc2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
DRD1 P21728 1/20 0.30
CYP1A2 P05177 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13840013 0.94 TDP1 (0.44) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL2085135 0.66 TDP1 (1.00) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL5028587 0.66 TDP1 (1.00) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL101 0.66 TDP1 (1.00) CYP3A4TDP1ESR1ESR2LMNA
Benzene SCHEMBL6890099 0.66 TDP1 (1.00) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL5076059 0.65 TDP1 (0.80) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL25384985 0.64 TDP1 (0.92) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL22558063 0.64 TDP1 (0.92) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL1195618 0.64 TDP1 (0.92) CYP3A4TDP1ESR1ESR2LMNA
SCHEMBL20582981 0.64 TDP1 (0.92) CYP3A4TDP1ESR1ESR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10858334-B2 Method for aerobic oxidative coupling of thiophenes with a ligand-supported palladium catalyst WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2020-12-08 US disclosed
US-20190210993-A1 Method for Aerobic Oxidative Coupling of Thiophenes with a Ligand-Supported Palladium Catalyst NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-07-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10858334-B2 Method for aerobic oxidative coupling of thiophenes with a ligand-supported palladium catalyst PPOX, TST, COX6C CYP3A4 164/4885TDP1 1835/4885ESR1 2454/4885
US-20190210993-A1 Method for Aerobic Oxidative Coupling of Thiophenes with a Ligand-Supported Palladium Catalyst PPOX, TST, COX6C CYP3A4 164/4885TDP1 1835/4885ESR1 2454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.