SCHEMBL21157461

SCHEMBL21157461

Cc1nc(-c2ccc(Oc3ccccc3)cc2)[nH]c1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.57
CHEK2 O96017 6/20 0.54
PIN1 Q13526 4/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
MAPK1 P28482 1/20 0.51
CASP1 P29466 1/20 0.51
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 2/20 0.47
GLA P06280 2/20 0.47
GAA P10253 2/20 0.47
HPGD P15428 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
GFER P55789 1/20 0.47
MAPK13 O15264 1/20 0.44
GCGR P47871 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21156706 0.86 DHODH (0.48) DHODHCHEK2PIN1CYP1A2CYP2C19
SCHEMBL8342056 0.79 MAPK1 (0.50) CHEK2PIN1CYP1A2CYP2C19MAPK1
SCHEMBL13309662 0.78 HRH3 (0.50) DHODHCHEK2PIN1MAPK1
SCHEMBL13982944 0.77 PIN1 (0.50) PIN1CYP1A2CYP2C19MAPK1CASP1
SCHEMBL4607219 0.75 ERCC1 (0.56) PIN1CYP1A2CYP2C19MAPK1CASP1
SCHEMBL11852911 0.74 DHODH (0.51) DHODHCHEK2PIN1MEN1KMT2A
SCHEMBL10552657 0.74 PKM (0.50) CHEK2CYP1A2CYP2C19KDM4EMEN1
SCHEMBL3760324 0.73 KDM4E (0.73) PIN1CYP1A2CYP2C19MAPK1CASP1
SCHEMBL30903772 0.73 MAPK13 (0.65) DHODHCHEK2MEN1GAAKMT2A
SCHEMBL504576 0.73 DHODH (0.68) DHODHCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2952513-B1 AZOLE BENZENE DERIVATIVE TEIJIN PHARMA LTD (JP) 2019-07-10 EP disclosed