SCHEMBL21158772

SCHEMBL21158772

CCc1nc(C)oc1C(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
LMNA P02545 3/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 3/20 0.36
STING1 Q86WV6 1/20 0.35
TSHR P16473 2/20 0.33
MEN1 O00255 2/20 0.33
USP2 O75604 2/20 0.33
POLB P06746 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177971 0.86 CYP1A2 (0.41) ALDH1A1LMNANPC1RAB9AKDM4E
SCHEMBL24562966 0.84 NPC1 (0.39) ALDH1A1LMNANPC1RAB9ARXFP1
SCHEMBL14125957 0.81 FBP1 (0.45) ALDH1A1LMNANPC1RAB9ARXFP1
SCHEMBL21158774 0.79 SMN1; SMN2 (0.37) ALDH1A1LMNANPC1RAB9AHSD17B10
SCHEMBL7140031 0.79 TARBP2 (0.44) ALDH1A1LMNANPC1RAB9AHSD17B10
SCHEMBL5013490 0.78 STING1 (0.36) ALDH1A1LMNANPC1RAB9AHSD17B10
SCHEMBL408193 0.77 ALDH1A1 (0.53) ALDH1A1LMNANPC1RAB9ANPSR1
SCHEMBL3826654 0.77 RNASEH1 (0.46) ALDH1A1LMNANPSR1HSD17B10KDM4E
SCHEMBL29689460 0.76 SMN1; SMN2 (0.31) ALDH1A1LMNANPC1RAB9AHSD17B10
Hydrochloric Acid SCHEMBL30823039 0.76 STING1 (0.35) ALDH1A1LMNANPC1RAB9AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111471056-B Macrocyclic immunomodulator 成都先导药物开发股份有限公司 2021-07-02 CN disclosed
CN-110016021-B Immunomodulator 成都先导药物开发股份有限公司 2021-05-07 CN disclosed
CN-111471056-A Macrocyclic immunomodulator 成都先导药物开发股份有限公司 2020-07-31 CN disclosed
WO-2020151682-A1 MACROCYCLIC IMMUNOMODULATOR 成都先导药物开发股份有限公司 2020-07-30 WO disclosed
WO-2019134707-A1 IMMUNOMODULATOR 成都先导药物开发股份有限公司 2019-07-11 WO disclosed