SCHEMBL21159436

SCHEMBL21159436

Nc1ncnc(N(N)Cc2ccc(F)cc2)c1N

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
MAP4K4 O95819 2/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
LMNA P02545 1/20 0.35
CSF1R P07333 1/20 0.34
AOC3 Q16853 1/20 0.34
RPS6KB1 P23443 2/20 0.34
IDO1 P14902 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
MAOB P27338 2/20 0.33
TP53 P04637 1/20 0.32
NSD2 O96028 1/20 0.32
NSD3 Q9BZ95 1/20 0.32
ELOVL1 Q9BW60 1/20 0.32
SLC2A1 P11166 1/20 0.32
PYCR1 P32322 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21159595 0.85 RAB9A (0.38) HTTESR1ESR2LMNACSF1R
SCHEMBL933733 0.68 ESR1 (0.57) ESR1ESR2AOC3IDO1LOXL2
SCHEMBL21159434 0.65 MAP4K4 (0.34) MAP4K4
SCHEMBL21090760 0.64 NUDT1 (0.35) HTTLMNA
SCHEMBL15597723 0.62 AOC3 (0.63) ESR1ESR2AOC3IDO1LOXL2
SCHEMBL2316376 0.62 CHEK1 (0.42) LMNATP53
SCHEMBL10664748 0.61 SMN1; SMN2 (0.42) HTTLMNA
SCHEMBL934572 0.61 BCL2A1 (0.51) ESR1ESR2AOC3LOXL2
SCHEMBL934617 0.61 ESR1 (0.49) ESR1ESR2AOC3LOXL2MAOB
SCHEMBL3906522 0.60 MPO (0.43) IDO1LOXL2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505171-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2019-07-03 EP disclosed