SCHEMBL21159574

SCHEMBL21159574

CN1CCCC(Nc2ncnc(N)c2NN)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 10/20 0.46
LRRK2 Q5S007 1/20 0.44
BPTF Q12830 1/20 0.40
BTK Q06187 1/20 0.39
NLRP3 Q96P20 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
PKM P14618 1/20 0.39
NFKB1 P19838 1/20 0.39
ADORA1 P30542 1/20 0.39
THPO P40225 1/20 0.39
PMP22 Q01453 1/20 0.39
HPGDS O60760 1/20 0.38
CHEK1 O14757 1/20 0.38
IL1B P01584 1/20 0.38
JAK3 P52333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21899550 0.78 BTK (0.44) KAT2BLRRK2BPTFBTKNLRP3
SCHEMBL27782780 0.73 HPGDS (0.69) BTKHPGDSJAK3
SCHEMBL3513711 0.73 KAT2B (0.44) KAT2BLRRK2BPTFNLRP3CHEK1
SCHEMBL25060362 0.70 BTK (0.59) KAT2BLRRK2BTKNLRP3CHEK1
SCHEMBL17622721 0.70 KAT2B (0.45) KAT2BLRRK2BPTFNLRP3ADORA1
SCHEMBL19649120 0.69 BTK (0.61) KAT2BBTK
SCHEMBL21705081 0.68 LRRK2 (0.54) LRRK2JAK3
SCHEMBL30973591 0.68 KAT2B (0.47) KAT2BBPTFNLRP3IL1B
SCHEMBL13226128 0.67 ROCK2 (0.52) KAT2BNLRP3CHEK1
SCHEMBL12676513 0.66 POLB (0.49) KAT2BBPTF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505171-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2019-07-03 EP disclosed