SCHEMBL21167441

SCHEMBL21167441

COc1ccc(Nc2cnc(N)c(N(N)Cc3ccc4ncccc4c3)n2)cn1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.41
PIK3CD O00329 9/20 0.41
PIK3CB P42338 9/20 0.41
PIK3CG P48736 9/20 0.41
MTOR P42345 2/20 0.40
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39
BRAF P15056 1/20 0.38
IGF1R P08069 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE10A Q9Y233 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29317449 0.84 ABCB1 (0.36) ABCB1ABCC1ABCG2NPC1
SCHEMBL24591153 0.83 GSK3A (0.39) MAPK10BRAFPDE10ANPC1RAB9A
SCHEMBL29314464 0.82 NPC1 (0.36) PDE10AABCB1ABCC1ABCG2NPC1
SCHEMBL21167442 0.82 PIK3CA (0.42) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL29314565 0.82 MET (0.34) BRAFIGF1RMEN1KMT2APDE10A
SCHEMBL22109644 0.81 ABCB1 (0.36) PIK3CABRAFIGF1RABCB1ABCC1
SCHEMBL22475873 0.80 BRAF (0.36) BRAFMEN1KMT2APDE10AABCB1
SCHEMBL24591158 0.80 MET (0.35) BRAFPDE10A
SCHEMBL24591103 0.80 GRM5 (0.36) ABCB1ABCC1ABCG2NPC1
SCHEMBL21167554 0.79 HDAC6 (0.34) PDE10ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed