SCHEMBL29314464

SCHEMBL29314464

CNP(NC)c1ccc(Nc2cnc(N)c(N(N)Cc3ccc4ncccc4c3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
DHFR P00374 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MET P08581 6/20 0.34
KLKB1 P03952 1/20 0.34
KLK1 P06870 1/20 0.34
HDAC3 O15379 1/20 0.33
EGFR P00533 1/20 0.32
TERT O14746 1/20 0.32
PDE10A Q9Y233 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CHKA P35790 1/20 0.32
PDK1 Q15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29317449 0.91 ABCB1 (0.36) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL29314565 0.87 MET (0.34) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL22109644 0.82 ABCB1 (0.36) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL21167441 0.82 PIK3CA (0.41) NPC1ABCB1ABCC1ABCG2PDE10A
SCHEMBL29314519 0.81 ABCB1 (0.33) ABCB1ABCC1ABCG2METKLKB1
SCHEMBL24591103 0.80 GRM5 (0.36) NPC1ABCB1ABCC1ABCG2MET
SCHEMBL29314533 0.79 ALOX5 (0.39) NPC1DHFRHDAC6KLKB1KLK1
SCHEMBL22475725 0.78 KDR (0.41) DHFRMETKLKB1KLK1HDAC3
SCHEMBL22475860 0.78 RECQL (0.35) ABCB1ABCC1ABCG2DHFRMET
SCHEMBL24591153 0.78 GSK3A (0.39) NPC1METKLKB1KLK1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3893872-B1 ORGANOPHOSPHORUS-SUBSTITUTED COMPOUNDS AS C-MET INHIBITORS AND THERAPEUTIC USES THEREOF BETA PHARMA INC (US) 2024-07-17 EP disclosed