SCHEMBL21173229

SCHEMBL21173229

C/C=C1\C(=O)c2ccc(C#N)cc2C1=C(C#N)C#N

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
CASP3 P42574 1/20 0.39
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
MALT1 Q9UDY8 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
EGFR P00533 2/20 0.33
RAD51 Q06609 1/20 0.33
ALK Q9UM73 3/20 0.32
PDPK1 O15530 1/20 0.32
MIF P14174 1/20 0.32
PDK2 Q15119 1/20 0.31
GSK3B P49841 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21173222 0.94 CASP3 (0.39) PKMMAPTALDH1A1GAACASP3
SCHEMBL21173228 0.83 USP8 (0.40) PKMMAPTALDH1A1GAAMEN1
SCHEMBL21173226 0.83 MAPT (0.39) PKMMAPTALDH1A1GAAMEN1
SCHEMBL25612614 0.81 USP8 (0.40) PKMMAPTALDH1A1GAAMEN1
SCHEMBL21173225 0.81 USP8 (0.40) PKMMAPTALDH1A1GAAMEN1
SCHEMBL2681526 0.80 S100A4 (0.42) PKMMAPTALDH1A1GAAMAOA
SCHEMBL2681524 0.80 S100A4 (0.42) PKMMAPTALDH1A1GAAMAOA
SCHEMBL16977316 0.80 S100A4 (0.42) PKMMAPTALDH1A1GAAMAOA
SCHEMBL24960484 0.79 MAPT (0.36) PKMMAPTALDH1A1GAAMEN1
SCHEMBL22544872 0.79 S100A4 (0.41) PKMMAPTALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019137354-A1 THIOPHENE-BASED FUSED AROMATIC SYSTEMS THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2019-07-18 WO disclosed