SCHEMBL21177474

SCHEMBL21177474

COc1ccc(-c2ccc3c(c2)C(=O)CC3)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.48
PBRM1 Q86U86 1/20 0.47
HSD17B1 P14061 1/20 0.46
PTGS2 P35354 1/20 0.45
HSD17B3 P37058 1/20 0.45
HDAC4 P56524 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
PDE4D Q08499 1/20 0.44
HRH3 Q9Y5N1 2/20 0.43
ALKBH3 Q96Q83 1/20 0.43
KDM4E B2RXH2 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1745460 0.87 HSD17B1 (0.63) HSD17B1PTGS2HSD17B3KDM4EHTT
SCHEMBL29392039 0.86 MAOB (0.54) BRD4PBRM1HRH3KDM4EHTT
SCHEMBL251842 0.86 MAOB (0.54) BRD4PBRM1HRH3KDM4EHTT
SCHEMBL5208267 0.81 BRD4 (0.55) BRD4PBRM1HSD17B1PTGS2PDE4D
SCHEMBL6130607 0.80 MAPK14 (0.56) KDM4EHTTMAOB
Butane SCHEMBL4688097 0.80 BRD4 (0.52) BRD4PBRM1HRH3KDM4EHTT
SCHEMBL7180348 0.79 MEN1 (0.56) BRD4PBRM1HSD17B1HSD17B3KDM4E
Acetic Acid SCHEMBL6934641 0.79 MAOB (0.51) BRD4PBRM1HRH3KDM4EHTT
SCHEMBL3010868 0.78 HSD17B1 (0.65) BRD4HSD17B1HTTMAOBALDH1A1
SCHEMBL27895 0.77 MAOB (0.67) BRD4HRH3MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141229-A1 COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF 上海怡立舍生物技术有限公司 2019-07-25 WO disclosed