SCHEMBL21178265

SCHEMBL21178265

Nc1cccc(CN2CCCC(O)C2)c1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.68
HTT P42858 2/20 0.56
KDM4E B2RXH2 3/20 0.52
POLB P06746 2/20 0.52
TSHR P16473 1/20 0.52
HPGD P15428 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ROCK2 O75116 4/20 0.49
CCR2 P41597 4/20 0.49
ROCK1 Q13464 4/20 0.49
CNR2 P34972 1/20 0.47
LTA4H P09960 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
PRMT6 Q96LA8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722397 0.91 ALDH1A1 (0.55) ALDH1A1HTTROCK2CCR2ROCK1
SCHEMBL4976833 0.86 ALDH1A1 (0.68) ALDH1A1HTTKDM4EPOLBTSHR
SCHEMBL3961183 0.82 CHRM2 (0.50) ALDH1A1HTTKDM4EPOLBROCK2
SCHEMBL1955800 0.82 ALDH1A1 (0.71) ALDH1A1HTTKDM4EPOLBTSHR
SCHEMBL1552926 0.82 ALDH1A1 (1.00) ALDH1A1HTTKDM4EPOLBTSHR
SCHEMBL1787570 0.82 ALDH1A1 (1.00) ALDH1A1HTTKDM4EPOLBTSHR
SCHEMBL5205368 0.82 ALDH1A1 (1.00) ALDH1A1HTTKDM4EPOLBTSHR
Methane SCHEMBL7287824 0.80 ALDH1A1 (0.97) ALDH1A1HTTKDM4EPOLBTSHR
Hydrochloric Acid SCHEMBL5343928 0.80 ALDH1A1 (0.97) ALDH1A1HTTKDM4EPOLBTSHR
SCHEMBL13242846 0.80 PRMT6 (0.62) ALDH1A1KDM4ESMN1; SMN2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3740207-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) Syros Pharmaceuticals, Inc. (US) 2020-11-25 EP disclosed
WO-2019143719-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS, INC. (US) 2019-07-25 WO disclosed