SCHEMBL2117860

SCHEMBL2117860

Cc1cc(S(=O)(=O)Nc2cc(-c3ccc(C#N)cn3)ccc2C)cs1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ACLY P53396 1/20 0.39
KDM1A O60341 2/20 0.38
MAOA P21397 2/20 0.38
SGK1 O00141 1/20 0.38
MAPT P10636 2/20 0.38
PIK3CA P42336 3/20 0.37
MTOR P42345 3/20 0.37
SLC22A12 Q96S37 1/20 0.37
CRBN Q96SW2 1/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2117688 0.86 ACLY (0.51) HSD11B1MEN1KMT2AACLYSGK1
SCHEMBL2122713 0.83 HSD11B1 (0.47) HSD11B1ACLYKDM1AMAOAMAPT
SCHEMBL2119034 0.83 TP53 (0.52) HSD11B1ACLYKDM1AMAOAMAPT
SCHEMBL2119726 0.83 KDM1A (0.48) HSD11B1ACLYKDM1AMAOAMAPT
SCHEMBL2118065 0.82 ALDH1A1 (0.40) HSD11B1MEN1KMT2AACLYKDM1A
SCHEMBL2117812 0.82 MAPT (0.48) MEN1KMT2AKDM1AMAOAMAPT
SCHEMBL2117136 0.82 TP53 (0.42) HSD11B1ACLYKDM1AMAOASGK1
SCHEMBL2119273 0.82 KDM4E (0.53) MEN1KMT2AMAPTPIK3CAMTOR
SCHEMBL2119673 0.81 ACLY (0.43) HSD11B1ACLYKDM1AMAOASGK1
SCHEMBL2122365 0.81 MAPT (0.43) HSD11B1ACLYKDM1AMAOASGK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120095012-A1 TOLUIDINE SULFONAMIDES AND THEIR USE ELARA PHARMACEUTICALS GMBH (DE) 2012-04-19 US disclosed
EP-2382190-A1 TOLUIDINE SULFONAMIDES AND THEIR USE AS-INHIBITORS European Molecular Biology Laboratory (EMBL) (DE) 2011-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095012-A1 TOLUIDINE SULFONAMIDES AND THEIR USE HIF1A, HIF1AN, EGLN3 HSD11B1 3376/4885MEN1 3143/4885KMT2A 290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.