SCHEMBL21185248

SCHEMBL21185248

CC#Cc1cccc2nc(CCC)n(C3CC3)c(=O)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 1/20 0.44
MAPK1 P28482 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE10A Q9Y233 2/20 0.38
PIK3CD O00329 3/20 0.37
PIK3R1 P27986 3/20 0.37
PIK3CG P48736 3/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
USP2 O75604 1/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2D6 P10635 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21185379 0.91 CRHBP (0.42) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL21185257 0.88 PIK3CD (0.48) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL21178215 0.84 PIK3CD (0.37) ALDH1A1LMNAHTTNPSR1MAPT
SCHEMBL21178492 0.83 NPSR1 (0.38) ALDH1A1LMNAMAPK1NPSR1MAPT
SCHEMBL16597161 0.82 ALDH1A1 (0.48) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL16597162 0.81 HSP90AB1 (0.49) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL16597166 0.81 ALDH1A1 (0.47) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL21174746 0.79 PIK3CD (0.46) PIK3CDPIK3R1PIK3CGPIK3CA
SCHEMBL21174744 0.79 PIK3CD (0.46) PIK3CDPIK3R1PIK3CGPIK3CA
SCHEMBL21185262 0.79 PIK3CD (0.49) PDE10APIK3CDPIK3R1PIK3CGCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143874-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2019-07-25 WO disclosed