SCHEMBL21187113

SCHEMBL21187113

N=C(Nc1ccc(Cl)cc1)N[C@H]1CC[C@@H](c2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.55
MAPT P10636 3/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
CNR1 P21554 2/20 0.45
ALDH1A1 P00352 3/20 0.43
EPHX1 P07099 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
POLB P06746 2/20 0.43
FPR1 P21462 2/20 0.42
FPR2 P25090 2/20 0.42
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187085 1.00 IDO1 (0.55) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL21187086 0.85 MEN1 (0.49) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL21187084 0.85 MEN1 (0.49) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL17730031 0.83 RAB9A (0.65) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL17730019 0.83 RAB9A (0.65) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL17730017 0.83 RAB9A (0.65) IDO1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL21187199 0.83 FPR1 (0.47) MAPTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL21187195 0.83 NPC1 (0.51) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL21187119 0.83 NPC1 (0.51) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL21187116 0.81 SMN1; SMN2 (0.39) IDO1NPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed