SCHEMBL21187116

SCHEMBL21187116

Cc1cc([C@H]2CC[C@H](NC(=N)Nc3ccc(Cl)cc3)CC2)cc(C)n1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
CYP2C19 P33261 2/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
EPHX1 P07099 1/20 0.39
CYP2C9 P11712 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ADRA2A P08913 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
HTR2B P41595 1/20 0.38
MCHR1 Q99705 1/20 0.38
IDO1 P14902 2/20 0.37
PROKR1 Q8TCW9 1/20 0.37
EPHX2 P34913 1/20 0.36
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187125 0.87 IDO1 (0.50) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187127 0.82 THRB (0.38) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187193 0.82 THRB (0.38) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187123 0.82 THRB (0.38) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187085 0.81 IDO1 (0.55) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187113 0.81 IDO1 (0.55) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21176926 0.79 NPC1 (0.37) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21176925 0.79 NPC1 (0.37) SMN1; SMN2CYP2C19NPC1ALDH1A1EPHX1
SCHEMBL21187199 0.78 FPR1 (0.47) SMN1; SMN2NPC1ALDH1A1EPHX1RAB9A
SCHEMBL17731108 0.76 IDO1 (0.55) SMN1; SMN2CYP2C9IDO1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed