SCHEMBL21187120

SCHEMBL21187120

Cc1ccncc1[C@H]1CC[C@@H](NC(=N)Nc2ccc(Cl)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.41
IDO1 P14902 3/20 0.41
NAMPT P43490 3/20 0.38
CYP2C9 P11712 3/20 0.37
CYP2C19 P33261 3/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
EPHX1 P07099 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP3A4 P08684 3/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2C8 P10632 1/20 0.35
TDO2 P48775 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAPK1 P28482 1/20 0.34
EPHX2 P34913 1/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187126 1.00 OPRL1 (0.41) OPRL1IDO1NAMPTCYP2C9CYP2C19
SCHEMBL21187138 0.80 IDO1 (0.50) IDO1CYP2C9CYP2C19RAB9ANPC1
SCHEMBL21187131 0.80 IDO1 (0.50) IDO1CYP2C9CYP2C19RAB9ANPC1
SCHEMBL21187116 0.75 SMN1; SMN2 (0.39) IDO1CYP2C9CYP2C19RAB9ANPC1
SCHEMBL21187125 0.75 IDO1 (0.50) IDO1NAMPTCYP2C9CYP2C19RAB9A
SCHEMBL21187113 0.73 IDO1 (0.55) IDO1CYP2C9CYP2C19RAB9ANPC1
SCHEMBL21187085 0.73 IDO1 (0.55) IDO1CYP2C9CYP2C19RAB9ANPC1
SCHEMBL10079573 0.72 OPRL1 (0.55) OPRL1IDO1
SCHEMBL11699099 0.72 EPHX1 (0.67) CYP2C9CYP2C19RAB9ANPC1ALDH1A1
SCHEMBL21187199 0.71 FPR1 (0.47) RAB9ANPC1ALDH1A1EPHX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed