SCHEMBL21187155

SCHEMBL21187155

COc1ccc(C2CCC(N/C(=N/I)Nc3ccc(Cl)cc3)CC2)nc1C

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.37
CHRM4 P08173 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
MEN1 O00255 3/20 0.35
THRB P10828 1/20 0.34
ALOX5 P09917 1/20 0.34
EPHX2 P34913 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
CYP2C9 P11712 2/20 0.33
MAPT P10636 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
EPHX1 P07099 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
CNR1 P21554 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187219 0.91 CHRM4 (0.37) KMT2ACHRM4L3MBTL1TDP1MEN1
SCHEMBL21187130 0.78 SMN1; SMN2 (0.39) KMT2AL3MBTL1TDP1MEN1THRB
SCHEMBL21187136 0.77 SMN1; SMN2 (0.40) KMT2AL3MBTL1TDP1MEN1THRB
SCHEMBL21187127 0.77 THRB (0.38) THRBEPHX2SMN1; SMN2CYP2C9NPC1
SCHEMBL21187193 0.77 THRB (0.38) THRBEPHX2SMN1; SMN2CYP2C9NPC1
SCHEMBL21187123 0.77 THRB (0.38) THRBEPHX2SMN1; SMN2CYP2C9NPC1
SCHEMBL21397172 0.69 MAPT (0.55) KMT2AL3MBTL1TDP1MEN1EPHX2
SCHEMBL21187213 0.68 NPC1 (0.48) KMT2AL3MBTL1MEN1EPHX2SMN1; SMN2
SCHEMBL22405862 0.66 ALDH1A1 (0.43) KMT2AL3MBTL1MEN1ALOX5SMN1; SMN2
SCHEMBL27316765 0.64 CACNA1B (0.39) L3MBTL1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed