SCHEMBL21187157

SCHEMBL21187157

Cc1nccc(C2CCC(NC(=N)Nc3cccc(F)c3)CC2)c1C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
KMT2A Q03164 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 2/20 0.41
GAA P10253 1/20 0.41
IDO1 P14902 3/20 0.40
TP53 P04637 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
HTR6 P50406 2/20 0.39
POLB P06746 2/20 0.39
EPHX2 P34913 1/20 0.38
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187153 0.86 NPC1 (0.45) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL21187166 0.82 MET (0.37) IDO1
SCHEMBL21187138 0.81 IDO1 (0.50) NPC1RAB9ASMN1; SMN2IDO1HTR6
SCHEMBL21187131 0.81 IDO1 (0.50) NPC1RAB9ASMN1; SMN2IDO1HTR6
SCHEMBL21187156 0.80 NPC1 (0.43) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL21187221 0.78 IDO1 (0.39) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL21187087 0.75 IDO1 (0.54) IDO1
SCHEMBL21187168 0.74 GRM4 (0.41) RAB9AIDO1
SCHEMBL21187159 0.72 IDO1 (0.37) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL23061556 0.69 IDO1 (0.50) IDO1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed