SCHEMBL21187153

SCHEMBL21187153

COc1cccc(NC(=N)NC2CCC(c3ccnc(C)c3C)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 5/20 0.42
NFKB1 P19838 1/20 0.42
CASP3 P42574 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
STAT1 P42224 1/20 0.41
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187156 0.90 NPC1 (0.43) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL21187157 0.86 NPC1 (0.41) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL21187166 0.82 MET (0.37) CASP3
SCHEMBL21187138 0.79 IDO1 (0.50) NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL21187131 0.79 IDO1 (0.50) NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL21187168 0.74 GRM4 (0.41) RAB9ACASP3GRM4
SCHEMBL21187221 0.72 IDO1 (0.39) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL6720800 0.69 TP53 (0.60) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL21187141 0.68 FPR1 (0.52) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL23061556 0.68 IDO1 (0.50) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed