SCHEMBL21189242

SCHEMBL21189242

COC(=O)N[C@H]1CCOc2c(C(=O)Nc3ccc(F)c(C(F)(F)F)c3)cccc21

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 8/20 0.47
PTGES O14684 3/20 0.46
KDR P35968 1/20 0.44
APOB P04114 4/20 0.44
MTTP P55157 4/20 0.44
GRM4 Q14833 1/20 0.41
SMO Q99835 2/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19973650 0.90 TRPV1 (0.48) TRPV1PTGESGRM4PTGS1
SCHEMBL19973651 0.90 TRPV1 (0.48) TRPV1PTGESGRM4PTGS1
SCHEMBL21189262 0.90 TP53 (0.42) TRPV1PTGESAPOBMTTP
SCHEMBL21189485 0.90 TP53 (0.42) TRPV1PTGESAPOBMTTP
SCHEMBL21189206 0.90 TP53 (0.42) TRPV1PTGESAPOBMTTP
SCHEMBL21189284 0.88 APOB (0.42) TRPV1PTGESAPOBMTTPSMO
SCHEMBL21189278 0.87 FADS1 (0.46) PTGESAPOBMTTP
SCHEMBL19973620 0.86 RXFP1 (0.51) PTGS1
SCHEMBL21189267 0.85 AKR1C3 (0.38) TRPV1PTGESAPOBMTTP
SCHEMBL21189281 0.85 LMNA (0.41) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11001564-B2 Substituted chromane-8-carboxamide compounds and analogues thereof, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2021-05-11 US disclosed
US-20190225593-A1 SUBSTITUTED CHROMANE-8-CARBOXAMIDE COMPOUNDS AND ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (CA) 2019-07-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190225593-A1 SUBSTITUTED CHROMANE-8-CARBOXAMIDE COMPOUNDS AND ANALOGUES THEREOF, AND METHODS USING SAME CBX8, HAVCR2, HCCS TRPV1 3647/4885PTGES 4518/4885KDR 4106/4885
US-11001564-B2 Substituted chromane-8-carboxamide compounds and analogues thereof, and methods using same CBX8, HAVCR2, HCCS TRPV1 3647/4885PTGES 4518/4885KDR 4106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.